Effect of estrogen and related compounds on the release of [3H]AEA from HUVECs preloaded with [3H]AEA
Sample . | [3H]AEA release, % control . |
---|---|
Control | 100* |
+100 nM E2 | 600 ± 60† |
+100 nM E2+100 nM TMX | 105 ± 10‡ |
+100 nM E2+100 nM ICI182780 | 580 ± 58† |
+100 nM E2+2 μM SR141716 | 520 ± 52† |
+100 nM E2+100 nM HU-210 | 950 ± 95†,2-153 |
+100 nM E2+2 μM CBD | 585 ± 58† |
+100 nM E2+2 μM CAPS | 600 ± 60† |
+100 nM E2+10 μM AM404 | 150 ± 15‡ |
+100 nM E2+400 μMl-NAME | 160 ± 16‡ |
+100 nM E2+50 μM EGTA-am | 150 ± 15‡ |
Sample . | [3H]AEA release, % control . |
---|---|
Control | 100* |
+100 nM E2 | 600 ± 60† |
+100 nM E2+100 nM TMX | 105 ± 10‡ |
+100 nM E2+100 nM ICI182780 | 580 ± 58† |
+100 nM E2+2 μM SR141716 | 520 ± 52† |
+100 nM E2+100 nM HU-210 | 950 ± 95†,2-153 |
+100 nM E2+2 μM CBD | 585 ± 58† |
+100 nM E2+2 μM CAPS | 600 ± 60† |
+100 nM E2+10 μM AM404 | 150 ± 15‡ |
+100 nM E2+400 μMl-NAME | 160 ± 16‡ |
+100 nM E2+50 μM EGTA-am | 150 ± 15‡ |