Agonists, antagonists, and inhibitors used in this investigation
Compound . | Action . | Reference . |
---|---|---|
Tamoxifen (TMX) | Estrogen receptor antagonist | 6 |
ICI182780 | Nuclear estrogen receptor antagonist | 6 |
HU-210 | Synthetic CB1 receptor agonist | 32 |
SR141716 | CB1 receptor antagonist | 32 |
SR144528 | CB2 receptor antagonist | 32 |
Cannabidiol (CBD) | Endothelial-type CB receptor antagonist | 33 |
Abnormal-CBD | Synthetic endothelial-type CB receptor agonist | 33 |
Capsazepine (CAPS) | Vanilloid receptor antagonist | 11 |
Capsaicin | Natural vanilloid receptor agonist | 11 |
l-NAME | NOS inhibitor | 24 |
AM404 | AMT inhibitor | 34 |
Suramin | PLD inhibitor | 35 |
ST638 | Tyrosine kinase/PLD inhibitor | 36 |
ATFMK | FAAH inhibitor | 20 |
ETYA | 15-LOX inhibitor | 30 |
Compound . | Action . | Reference . |
---|---|---|
Tamoxifen (TMX) | Estrogen receptor antagonist | 6 |
ICI182780 | Nuclear estrogen receptor antagonist | 6 |
HU-210 | Synthetic CB1 receptor agonist | 32 |
SR141716 | CB1 receptor antagonist | 32 |
SR144528 | CB2 receptor antagonist | 32 |
Cannabidiol (CBD) | Endothelial-type CB receptor antagonist | 33 |
Abnormal-CBD | Synthetic endothelial-type CB receptor agonist | 33 |
Capsazepine (CAPS) | Vanilloid receptor antagonist | 11 |
Capsaicin | Natural vanilloid receptor agonist | 11 |
l-NAME | NOS inhibitor | 24 |
AM404 | AMT inhibitor | 34 |
Suramin | PLD inhibitor | 35 |
ST638 | Tyrosine kinase/PLD inhibitor | 36 |
ATFMK | FAAH inhibitor | 20 |
ETYA | 15-LOX inhibitor | 30 |